Event Description
December 2024 - 1034th Monthly Meeting of NESACS: Contemporary Methods in Medicinal Chemistry Symposium
This meeting will be hosted by Takeda in Cambridge, MA
Registration is required and ends at 11:30 PM on December 5, 2024
Registration is required and ends at 11:30 PM on December 5, 2024 Registration is required and ends at 11:30 PM on December 5, 2024 Thursday – December 12th, 2024
Takeda- 35 Lansdowne Street, Cambridge Massachusetts 02139
3:15 pm Welcome: Raj Rajur, Medicinal Chemistry Program Chair - CreaGen, Woburn, MA
3:20 pm - Introductory Remarks from Takeda
3:30 pm – 4:00 pm - Presentation: Ryan Kerrigan - Novartis
Ryan Kerrigan - Ryan Kerrigan - Title: “First-in-Class Molecular Glue Degraders of the WIZ Transcription Factor to Treat Sickle Cell Disease”
Title: “First-in-Class Molecular Glue Degraders of the WIZ Transcription Factor to Treat Sickle Cell Disease” Title: “First-in-Class Molecular Glue Degraders of the WIZ Transcription Factor to Treat Sickle Cell Disease” 4:00 pm – 4:45 pm - Presentation: Michelle Garnsey - Pfizer
Michelle Garnsey Michelle Garnsey Title: "Discovery of SARS-CoV-2 papain-like protease (PLpro) inhibitors with efficacy in a murine infection model"
4:45 - 5:00 pm - Break
5:00 pm – 5:45 pm - Presentation: Derun Li - Nimbus
Derun Li Derun Li Title: "Designing Selective WRN Covalent Inhibitors from Non-Covalent Binders"
5:45 pm - 6:30 pm - Presentation: Brandon Vara – Merck
Brandon Vara Brandon Vara Title: "Discovery of MK-4424: a Potent, Exquisitely Selective, and CNS-penetrant RIPK1 Type-III Inhibitor to Treat Neurodegeneration"
6:45 pm – 8:30 pm Dinner
THE PUBLIC IS INVITED - RESERVATIONS ARE REQUIRED
THE PUBLIC IS INVITED - RESERVATIONS ARE REQUIRED THE PUBLIC IS INVITED - RESERVATIONS ARE REQUIRED YOU MUST REGISTER IN ADVANCE TO ATTEND THE SYMPOSIUM: THERE IS NO REGISTRATION FEE TO ATTEND THE SYMPOSIUM, DINNER RESERVATIONS ARE REQUIRED.
YOU MUST REGISTER IN ADVANCE TO ATTEND THE SYMPOSIUM: THERE IS NO REGISTRATION FEE YOU MUST REGISTER IN ADVANCE TO ATTEND THE SYMPOSIUM: THERE IS NO REGISTRATION FEE YOU MUST REGISTER IN ADVANCE TO ATTEND THE SYMPOSIUM: THERE IS NO REGISTRATION FEE TO ATTEND THE SYMPOSIUM, DINNER RESERVATIONS ARE REQUIRED. TO ATTEND THE SYMPOSIUM, DINNER RESERVATIONS ARE REQUIRED. TO ATTEND THE SYMPOSIUM, DINNER RESERVATIONS ARE REQUIRED. Please use google map: 35 Lansdowne Street, Cambridge Massachusetts 02139.
Please use google map: Please use google map: MBTA closest stop is Central Square on the red line. Bus lines 1 and 2.
MBTA closest stop is Central Square on the red line. Bus lines 1 and 2. MBTA closest stop is Central Square on the red line. Bus lines 1 and 2. Parking is available at 10 Green St., directly across from the symposium entrance. Parking is free if validated at the entrance desk.
Parking is available at 10 Green St., directly across from the symposium entrance. Parking is free if validated at the entrance desk. Parking is available at 10 Green St., directly across from the symposium entrance. Parking is free if validated at the entrance desk. Attendees will need to enter via the back entrance to the building, which is located on Green St.
Attendees will need to enter via the back entrance to the building, which is located on Green St. Attendees will need to enter via the back entrance to the building, which is located on Green St. Registration or other questions? Please contact: Jaison by email at jason.beiger@takeda.com or Raj Rajur rrajur@creageninc.com
Registration or other questions? Please contact: Jaison by email at Registration or other questions? Please contact: Jaison by email at jason.beiger@takeda.com or Raj Rajur or Raj Rajur rrajur@creageninc.com Organizing Committee:
Mark Ashwell; Brian. Aquila; Blaise Lippa; Andrew Scholte; Peter Fuller; Michelle Lamb; Silvana Leit; Melissa Grenier-Davies; Paul Scola; Lauren Monovich; Jason Beiger; Paul Greenspan; Raj Rajur
Mark Ashwell; Brian. Aquila; Blaise Lippa; Andrew Scholte; Peter Fuller; Michelle Lamb; Silvana Leit; Melissa Grenier-Davies; Paul Scola; Lauren Monovich; Jason Beiger; Paul Greenspan; Raj Rajur Mark Ashwell; Brian. Aquila; Blaise Lippa; Andrew Scholte; Peter Fuller; Michelle Lamb; Silvana Leit; Melissa Grenier-Davies; Paul Scola; Lauren Monovich; Jason Beiger; Paul Greenspan; Raj Rajur Mark Ashwell; Brian. Aquila; Blaise Lippa; Andrew Scholte; Peter Fuller; Michelle Lamb; Silvana Leit; Melissa Grenier-Davies; Paul Scola; Lauren Monovich; Jason Beiger; Paul Greenspan; Raj Rajur
This meeting will be hosted by Takeda in Cambridge, MA
Registration is required and ends at 11:30 PM on December 5, 2024
Registration is required and ends at 11:30 PM on December 5, 2024 Registration is required and ends at 11:30 PM on December 5, 2024 Thursday – December 12th, 2024
Takeda- 35 Lansdowne Street, Cambridge Massachusetts 02139
3:15 pm Welcome: Raj Rajur, Medicinal Chemistry Program Chair - CreaGen, Woburn, MA
3:20 pm - Introductory Remarks from Takeda
3:30 pm – 4:00 pm - Presentation: Ryan Kerrigan - Novartis
Ryan Kerrigan - Ryan Kerrigan - Title: “First-in-Class Molecular Glue Degraders of the WIZ Transcription Factor to Treat Sickle Cell Disease”
Title: “First-in-Class Molecular Glue Degraders of the WIZ Transcription Factor to Treat Sickle Cell Disease” Title: “First-in-Class Molecular Glue Degraders of the WIZ Transcription Factor to Treat Sickle Cell Disease” 4:00 pm – 4:45 pm - Presentation: Michelle Garnsey - Pfizer
Michelle Garnsey Michelle Garnsey Title: "Discovery of SARS-CoV-2 papain-like protease (PLpro) inhibitors with efficacy in a murine infection model"
4:45 - 5:00 pm - Break
5:00 pm – 5:45 pm - Presentation: Derun Li - Nimbus
Derun Li Derun Li Title: "Designing Selective WRN Covalent Inhibitors from Non-Covalent Binders"
5:45 pm - 6:30 pm - Presentation: Brandon Vara – Merck
Brandon Vara Brandon Vara Title: "Discovery of MK-4424: a Potent, Exquisitely Selective, and CNS-penetrant RIPK1 Type-III Inhibitor to Treat Neurodegeneration"
6:45 pm – 8:30 pm Dinner
THE PUBLIC IS INVITED - RESERVATIONS ARE REQUIRED
THE PUBLIC IS INVITED - RESERVATIONS ARE REQUIRED THE PUBLIC IS INVITED - RESERVATIONS ARE REQUIRED YOU MUST REGISTER IN ADVANCE TO ATTEND THE SYMPOSIUM: THERE IS NO REGISTRATION FEE TO ATTEND THE SYMPOSIUM, DINNER RESERVATIONS ARE REQUIRED.
YOU MUST REGISTER IN ADVANCE TO ATTEND THE SYMPOSIUM: THERE IS NO REGISTRATION FEE YOU MUST REGISTER IN ADVANCE TO ATTEND THE SYMPOSIUM: THERE IS NO REGISTRATION FEE YOU MUST REGISTER IN ADVANCE TO ATTEND THE SYMPOSIUM: THERE IS NO REGISTRATION FEE TO ATTEND THE SYMPOSIUM, DINNER RESERVATIONS ARE REQUIRED. TO ATTEND THE SYMPOSIUM, DINNER RESERVATIONS ARE REQUIRED. TO ATTEND THE SYMPOSIUM, DINNER RESERVATIONS ARE REQUIRED. Please use google map: 35 Lansdowne Street, Cambridge Massachusetts 02139.
Please use google map: Please use google map: MBTA closest stop is Central Square on the red line. Bus lines 1 and 2.
MBTA closest stop is Central Square on the red line. Bus lines 1 and 2. MBTA closest stop is Central Square on the red line. Bus lines 1 and 2. Parking is available at 10 Green St., directly across from the symposium entrance. Parking is free if validated at the entrance desk.
Parking is available at 10 Green St., directly across from the symposium entrance. Parking is free if validated at the entrance desk. Parking is available at 10 Green St., directly across from the symposium entrance. Parking is free if validated at the entrance desk. Attendees will need to enter via the back entrance to the building, which is located on Green St.
Attendees will need to enter via the back entrance to the building, which is located on Green St. Attendees will need to enter via the back entrance to the building, which is located on Green St. Registration or other questions? Please contact: Jaison by email at jason.beiger@takeda.com or Raj Rajur rrajur@creageninc.com
Registration or other questions? Please contact: Jaison by email at Registration or other questions? Please contact: Jaison by email at jason.beiger@takeda.com or Raj Rajur or Raj Rajur rrajur@creageninc.com Organizing Committee:
Mark Ashwell; Brian. Aquila; Blaise Lippa; Andrew Scholte; Peter Fuller; Michelle Lamb; Silvana Leit; Melissa Grenier-Davies; Paul Scola; Lauren Monovich; Jason Beiger; Paul Greenspan; Raj Rajur
Mark Ashwell; Brian. Aquila; Blaise Lippa; Andrew Scholte; Peter Fuller; Michelle Lamb; Silvana Leit; Melissa Grenier-Davies; Paul Scola; Lauren Monovich; Jason Beiger; Paul Greenspan; Raj Rajur Mark Ashwell; Brian. Aquila; Blaise Lippa; Andrew Scholte; Peter Fuller; Michelle Lamb; Silvana Leit; Melissa Grenier-Davies; Paul Scola; Lauren Monovich; Jason Beiger; Paul Greenspan; Raj Rajur Mark Ashwell; Brian. Aquila; Blaise Lippa; Andrew Scholte; Peter Fuller; Michelle Lamb; Silvana Leit; Melissa Grenier-Davies; Paul Scola; Lauren Monovich; Jason Beiger; Paul Greenspan; Raj Rajur
Event Location
Tags
science-innovationsustainability-conferenceeducationrobotics-aitech
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